I-Megace isetshenziselwa ukugqugquzela ukudla kubantu abane-AIDS nomdlavuza
I-Megace (i-megestrol acetate) inikezwa abantu abagulayo kakhulu ngesifo somdlavuza webele, umdlavuza we-endometrial noma i-AIDS. Lesi sidakamizwa sinikezwa ukukhulisa ukudla nokuzuza kwesisindo. Kulezi ziguli ezigula kakhulu futhi ezibekwe i-Megace, imiphumela ye-hormone yalesi sidakamizwa ingathuthukisa futhi ibangele ukwanda kwenhlalakahle, futhi.
Ngezinye izikhathi abantu asebekhulile nabangaphansi kwamandla banqunywe i-Megace, kodwa ukusebenza kwalesi sidakamizwa kubantu asebekhulile akuqinisekisiwe.
Iningi locwaningi lweMegace libandakanya labo abanomdlavuza noma i-AIDS.
I-Megace i-endocrine-i-agent ye-metabolic ne-hormone yokwenziwa. Ngenxa yokuthi i-Megace iyinhlangano ye-hormone yokwenziwa, inezimo ezihlukahlukene ezimbi ezibandakanya izinhlelo eziningi zomzimba ezihamba kuwo wonke umzimba.
Inqubo yesenzo
I-megace noma i-megestrol acetate yi-progestin yokwenziwa ene-antiestrogen futhi ingase isebenze i-endometrium noma i-lining kwesibeletho. Ngokuqondile, i-Megace iphazamisa umjikelezo we-estrogen-receptor futhi kucatshangwa ukuthi ibangele igwebu le-pituitary ebuchosheni (elifanekiselwe kulesi sihloko). I-pituitary gland ifihla ama-hormone ehlasela imisipha yakho, izinso, nezitho ezihlukahlukene. Abanye ochwepheshe bakholelwa ukuthi i-Megace ikhuthaza ukudla ngenxa yomphumela wayo emzimbeni we-metabolism (i-cytokines yamathambo).
Izimpawu zomtholampilo ze-Megace
I-Megace inikezwa ku-:
- ukukhulula ukuhlupheka okubangelwa umdlavuza we-endometrial noma umdlavuza webele;
- ukwandisa ukudla nokuyeka ukulahlekelwa isisindo kubantu abane-AIDS nomdlavuza (i-cachexia)
- ukwandisa ukondla umdlavuza wesi-prostate
- ukukhuthaza isimo sengqondo kubantu abane-AIDS nomdlavuza
- ukuhlinzeka ngemithi ye-hormone ye-endometrial nesifo somdlavuza webele
Njengoba kushiwo ngaphambili, akukho ukusekelwa okusekelwe ebufakazini bokusetshenziswa kweMegace njengokwelashwa kokulahlekelwa yilaba bantu asebekhulile.
Imiphumela emibi ye-Megace
I-Megace ayikho ukuxhumana nezinye izidakamizwa.
Kodwa-ke, i-Megace inezinyathelo zomtholampilo eziningi futhi ingaphazamisa impilo nenhlalakahle ngezindlela ezihlukahlukene, ohlwini olulandelayo, kungenzeka imiphumela emibi ye-Megace ilandelwa ukukhula okulinganisiwe.
- umfutho wegazi ophezulu (amaphesenti angu-4 kuya kwangu-8)
- ubuhlungu besifuba (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- ama-palpitations (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- i-headache (amaphesenti amathathu kuya kwangu-10)
- ukulala (amaphesenti angu-1 kuya kwangu-6)
- ukucindezeleka (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- ukuphelelwa yisifo senhliziyo noma ubuthakathaka benhliziyo (amaphesenti angu-1 amaphesenti amathathu)
- ukuqhuma kwesikhumba (amaphesenti ayisithupha kuya kwamaphesenti angu-12)
- i-pruritis noma isikhumba sesikhumba (amaphesenti angu-1 kuya ku-3 amaphesenti)
- i-hyperglycemia noma ushukela ophezulu (amaphesenti angu-6)
- ukukhuliswa kwesifuba noma i-gynecomastia (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- isifo sohudo (amaphesenti angu-10 futhi alingana ne-placebo)
- ukuqotshwa (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- ukungabi namandla (amaphesenti angu-4 kuya kuma-14 amaphesenti)
- ukungabikho komchamo (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- ukutheleleka (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- izinkinga zamehlo (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- ukukhwehlela (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- umkhuhlane (amaphesenti angu-1 kuya kwangu-6)
- ukutheleleka (amaphesenti angu-1 kuya kwamaphesenti amathathu)
- isibindi esikhulu noma i-hepatomegaly (amaphesenti angu-1 kuya kwamaphesenti amathathu)
Inothi, i-Megace akufanele ithathwe ngesikhathi sokukhulelwa futhi ingalimaza ingane.
Ngafaka izinto eziningi kulolu hlu ukufakazela iphuzu: I-Megace iyi-hormone, futhi abantu abaningi abathatha ama-hormone bazobhekana nemiphumela emibi emibi.
Ukwelapha ama-hormone kufanele kucatshangelwe ngokucophelela futhi ngezinye izikhathi kungacindezela izifo zenhliziyo noma kungabangela ukucindezeleka okukhulu. Ngenxa yalesi sizathu, i-Megace iyisisetshenziswa esingcono kakhulu esilondolozwe abantu ekunakekelweni kokugcina, hhayi abantu asebekhulile abadinga isisindo.
Uma uthatha i-Megace futhi uzwa ubuhlungu besifuba, isicanucanu, ukuhlanza, ukuvuthwa okuvamile, ubuhlungu bomlenze, noma yini enye eyenza uzizwe unesihluku, qiniseka ukuyeka ukusebenzisa imithi bese ubona udokotela ngokushesha. Uma kunesidingo, shayela izinsizakalo eziphuthumayo.
I-Megace itholakala kwifomu yomlomo njengokubili ukumiswa kanye nephilisi. Kukhona izinguqulo ezishibhile zama generic zale mithi etholakalayo.
Ngokuya komhlinzeki kanye nokubukwa kwezwe lokubekezela, isigxila esisodwa ku-Megace kwiziguli ezigugile yi-marijuana yezokwelapha.
Khetha Imithombo
Ukubukeza Komkhaya Ukuhlolwa Nokubukwa KweBhodi, Uhlobo Lwemithathu ngu-M Graber noJ Wilber olwanyatheliswa ngo-2012.
Izinkomba Zezidakamizwa ZakwaMosby, ezokuPhathwa kwezeMpilo , Ukushicilelwa kwesibili ezanyatheliswa ngo-2010.