Izidakamizwa ze-Antithyroid ezisetshenziselwa ukuphatha izifo zamathuna kanye ne-Hyperthyroidism
Izidakamizwa ze-Antithyroid - nazo ezibizwa ngokuthi ama-thioamide - ziyimithi ephathwa nge-thyroid engapheli (hyperthyroidism) ngokuvimbela ikhono legciwane le-thyroid lokukhiqiza i-hormone ye-thyroid. Lapho ukwelashwa ngokweqile, okuvame ukuphumela esimweni sokuzimela esibizwa ngokuthi yi-Graves's disease, kubalulekile ukunciphisa ukukhiqizwa ngokweqile kwamahomoni wegciwane, ikakhulukazi ama hormone thyroxine (T4) ne-triiodothyronine (T3).
Izidakamizwa ze-Antithyroid zenza ngokwenza kube nzima ngomzimba ukusebenzisa iodine, ngaleyo ndlela kuvimbele ukwakhiwa kwamahomoni wegciwane emgodini.
I-Antithyroid yokwelapha izidakamizwa ingenye yezokwelapha ze-hyperthyroidism ne-Graves's disease. Ezinye izindlela zokwelashwa zibandakanya ukususwa kwe-iodine ye-iodine (RAI) nokususwa kokuhlinzwa konke noma ingxenye yengane ye- thyroid .
Kunezidakamizwa ezimbili ezibalulekile ze-antithyroid okwamanje etholakalayo e-United States: propylthiouracil (PTU) ne-methimazole. E-United States, i-methimazole ithathwa njengesidakamizwa esithandwayo se-antithyroid ezimweni eziningi.
I-Methimazole, ngezinye izikhathi ebizwa ngokuthi i-thiamazole, ivimbela i-thyroid ngokusebenzisa i- iodine ukukhiqiza i-hormone yegciwane. Ngokuvamile kuthathwa njengomthamo kanye ngosuku.
Isidakamizwa sisetshenziswa emhlabeni jikelele. E-United States, i-Tapazole yiyona yedwa igama lomuthi we-antithyroid yezidakamizwa methimazole. Kukhona inani labakhiqizi abajwayelekile bama-methimazole.
I-Tapazole
I-Tapazole yigama le- methimazole , umuthi we-antithyroid owenziwe yi-King Pharmaceuticals, Inc. I-FDA evunyelwe iTapazole ngo-2000.
I-Tapazole Izithako : i-methimazole USP; i-lactose monohydrate; i-magnesium stearate; isitashi (ummbila); isitashi se-pregelatinized; kanye ne-talc.
Amandla atholakalayo : 5 mg no-10 mg
I-Generic Methimazole (ngu-Sandoz)
USandoz, ilungu le-Novartis Group of Companies, wenza i-methimazole ejwayelekile. Yamukelwa yi-FDA ngo-2001.
I-Sandoz Methimazole Izithako: i- methimazole USP; i-lactose monohydrate; i-magnesium stearate; isitashi (ummbila); kanye ne-talc.
Amandla atholakalayo: 5 mg no-10 mg
I-Generic Methimazole (yi-Cedar Pharmaceuticals LLC)
Abakhiqizi beCedar Pharmaceuticals LLC i-methimazole ejwayelekile eyenziwa yi-United Research Laboratories. Imvume ye-FDA itholwe ngo-2005.
I-Cedar Pharmaceuticals Methimazole Izithako: i- methimazole USP; i-actose monohydrate; i-magnesium stearate; i-starch isitashi; kanye ne-talc.
Amandla atholakalayo: 5 mg, 10 mg, 15 mg, 20 mg
I-Generic Methimazole (yi-Activis Totowa)
I-Activis Totowa LLC abakhiqizi be-generic methimazole ne-FDA imvume yatholwa ngo-2007.
I-activis yama-malamazole Izithako methimazole USP; i-lactose monohydrate; i-magnesium stearate; isitashi esandulele; kanye ne-talc.
Amandla atholakalayo: 5 mg no-10 mg
I-Generic Methimazole (yi-Caraco Pharmaceutical Laboratories)
I-Caraco Pharmaceutical Laboratories, Ltd yakha i-methimazole ejwayelekile eyenziwe yi-FDA ngo-2007.
I-Caraco Methimazole Izithako: i- methimazole USP; i-lactose monohydrate; i-povidone; i-talc; croscarmellose; i-magnesium stearate; kanye nesitashi samabele.
Amandla atholakala: 5mg no-10mg
I-Generic Methimazole (yi-Par Pharmaceutical Companies)
Ama-Pharmaceutical Companies akhiqiza i-methimazole ejwayelekile.
Izithako: i- methimazole USP; i-lactose monohydrate; i-magnesium stearate; isitashi sommbila; kanye ne-talc.
Amandla atholakalayo: 5 mg no-10 mg
Imithombo:
I-Med Med, i-US Food and Drug Administration Medication Database.
I-FDA Ukuphepha Kokuphepha Kwezidakamizwa: Isixwayiso Esisha Sokuxwayiswa Kwesibindi Esibi Ukulimala Nge-Propylthiouracil, ngo-Ephreli 21, 2010
Ross, Douglas MD, "Ulwazi lokubekezela: izidakamizwa ze-Antithyroid," UpToDate . Kugcine ukubuyekezwa: Novemba 13, 2009
Ukubika okungeziwe ngu: Leslie Blumenberg