I-Muscle Relaxer
I-Robaxin (i-Methocarbamol) iboniswa njengendlela yokuphumula yokuphumula, ukwelashwa ngokomzimba, nezinye izinyathelo zokukhululeka kokungahambi kahle ezihambisana nezimo ezibucayi, ezibuhlungu zomshukela. Imodi yesenzo se-methocarbamol ayizange ibonakale ngokucacile, kodwa ingahle ihlobene nezindawo zayo zokuvimbela. I-Robaxin ayiphumuli ngokuqondile imisipha yamathambo emadodeni.
Ukungafani
I-Robaxin iphikisana neziguli ezixhumene ne-methocarbamol noma kunoma yiziphi izingxenye zethebhulethi.
Izixwayiso
Njengoba i-methocarbamol ingaba nomphumela ovamile we-CNS ocindezelayo, iziguli ezithola i-Robaxin kufanele zixwayiswe ngemiphumela ehlanganisiwe ngotshwala nezinye izidakamizwa ze-CNS.
Ukusetshenziswa okuphephile kweRobaxin akuzange kusungulwe ngokuphathelene nemiphumela emibi engenzeka ekuthuthukiseni ingane. Kube khona imibiko yokukhubazeka kokubeletha nokuzalwa okungenasifo esilandelayo ngokulandela ukuvezwa kwe-utero kumethocarbamol. Ngakho-ke, i-Robaxin akufanele isetshenziswe kulabo besifazane abakhulelwe noma abakhulelwe ikakhulukazi ngesikhathi sokukhulelwa ngaphambi kokuba kutholakale isahlulelo sodokotela izinzuzo ezingaphezu kwezingozi ezikhona.
I-Robaxin ingaphazamisa amakhono engqondo kanye / noma emzimbeni adingekayo ekwenzeni imisebenzi enobungozi, njengemishini yokusebenza noma ukushayela imoto.
Ukuqapha
Iziguli kufanele ziqaphele ukuthi i-Robaxin ingabangela ukulala noma isizungu, okungase kuphazamise ikhono labo lokusebenzisa izimoto noma imishini.
Ngenxa yokuthi i-Robaxin ingase ibe nomthelela ovamile we-CNS-ecindezelayo, iziguli kufanele zixwayiswe ngemiphumela ehlangene ngotshwala nezinye izidakamizwa ze-CNS.
Ukusabela okubi
Ukusabela okubi kubikwa ukuthi kuhambisana nokuphathwa kwe-methocarbamol kufaka:
- Umzimba wonke: Ukusabela kwe-Anaphylactic, i-edema yama-angioneurotic, imfiva, ikhanda
- Isimo senhliziyo: I- Bradycardia, i-flushing, i-hypotension, i-syncope, i-thrombophlebitis
- I-digestive system : i- Dyspepsia, i-jaundice (kufaka phakathi i-jaundice ye-cholestatic), isisulu sokunambitheka nokuhlanza
- Uhlelo lweHemic and lymphatic: Leukopenia
- Amasosha omzimba : Ukuphendula kwe-Hypersensitivity
- Uhlelo lwezinzwa : i- Amnesia, ukudideka, i-diplopia, isizungu noma ukukhanya okuncane, ukulala, ukulala, ukungazinzi, ukungahambisani kahle kwemisipha, i-nystagmus, i-sedation, ukuhlukunyezwa (kufaka phakathi i-mal grand), i-vertigo
- Isikhumba nezinzwa ezikhethekile: Umbono ophukile, i-conjunctivitis, ukuminyanisa kwesisu, ukunambitheka kwe-metallic, i-pruritus, i-rash, i-urticaria
Ukusebenzisana kwezidakamizwa kanye nelebhu
I-Robaxin ingavimbela umphumela we-pyridostigmine bromide. Ngakho-ke, i-Robaxin kufanele isetshenziswe ngokucophelela ezigulini ezine-myasthenia gravis ezithola ama-anticholinesterase agents.
I-Methocarbamol ingabangela ukuphazamiseka kombala kwezinye izivivinyo zokuhlolwa kwe-5-hydroxyindoleacetic acid.
I-Carcinogenesis, i-Mutagenesis, Ukulimala kokuzala
Izifundo zesikhathi eside ukuze zihlolwe ikhono le-carcinogenic ye-Robaxin azenzanga. Azikho ucwaningo olwenziwe ukuze kuhlolwe umphumela weRobaxin on mutagenesis noma amandla awo okulimaza ukuzala.
Ukukhulelwa
Izifundo zokukhiqiza izilwane azizange zenziwe nge-methocarbamol.
Ayaziwa ukuthi ngabe i-methocarbamol ingabangela ukulimala komntwana uma iphathwe owesifazane okhulelwe noma ingathinta umthamo wokukhiqiza. I-Robaxin kufanele inikwe owesifazane okhulelwe kuphela uma kudingeka ngokucacile.
Ukusetshenziswa okuphephile kweRobaxin akuzange kusungulwe ngokuphathelene nemiphumela emibi engenzeka ekuthuthukiseni ingane. Kube khona imibiko yokukhubazeka kokubeletha nokuzalwa okungenasifo esilandelayo ngokulandela ukuvezwa kwe-utero kumethocarbamol. Ngakho-ke, i-Robaxin akufanele isetshenziswe kulabo besifazane abakhulelwe noma abakhulelwe ikakhulukazi ngesikhathi sokukhulelwa ngaphambi kokuba kukhishwe isazi izinzuzo ezingase zibe ngaphezu kwezingozi ezikhona.
Omama Abahlengikazi
I-Methocarbamol kanye / noma i-metabolite yayo idonswa ngobisi lwezinja; Kodwa-ke, awaziwa ukuthi i-methocarbamol noma i-metabolite yayo isetshenziselwa ubisi lomuntu. Ngenxa yokuthi izidakamizwa eziningi zidonswa ubisi lomuntu, ukuqaphela kufanele kusetshenziswe lapho uRobaxin enikezwa owesifazane onesihlengikazi.
Ukusetshenziswa kwezingane
Ukuphepha nokusebenza kwe-Robaxin ngeziguli ezingaphansi kwezingane ezingaphansi kweminyaka engu-16 azange zisungulwe.
I-Overdosage
Ukwaziswa okulinganiselwe kuyatholakala ngobunobuthi obukhulu be-methocarbamol. Ukudlula ngokweqile kwe-methocarbamol kuvame ukuhambisana notshwala noma ezinye izidakamizwa ze-CNS futhi kufaka phakathi izimpawu ezilandelayo:
- isiyaluyalu
- ukulala
- umbono ongenalutho
- hypotension
- ukuhlukunyezwa
- i-coma
Ekuhlangenwe nakho kokuthungatha, ukushona kuye kwabikwa ngokweqile kwe-methocarbamol yedwa noma phambi kwezinye izidakamizwa ze-CNS, izidakamizwa eziphuza utshwala noma zengqondo. Ukuphathwa kokudlula ngokweqile kubandakanya ukwelashwa okuphawulekayo nokusekela.
Gcina i-Robaxin endaweni yokushisa egumbini elilawulwayo, phakathi kuka-20 ° C no-25 ° C (68 ° F no-77 ° F).
Umthombo:
Ukuphathwa Kwezokudla Nezidakamizwa zase-US, i-NDA 11-011 / S-070/071