Imithi yomlomo ebizwa nge-Januvia (sitagliptin phosphate) ivunyiwe yi-US Food and Drug Administration yokuphatha uhlobo lwesifo sikashukela . Ngowokuqala ekilasini lemithi ebizwa ngokuthi i-DPP-4 inhibitors. UJanuya unciphisa amazinga kashukela egazi ngokuvimbela i-enzyme eyaziwa njenge-dipeptidyl peptidase IV noma i-DPP-4.
Uhlobo Luni Oluyisifo Sikashukela?
Uhlobo lwesifo sikashukela sesi-2, esaziwa ngokuthi isifo sikashukela esingabadala noma esingaxhaswanga yi-noninsulin, yisifo esingapheliyo esithinta indlela umzimba wakho ubeka ngayo ushukela (i-glucose), umthombo obalulekile womzimba wakho.
Nge-type 2 yesifo sikashukela, umzimba wakho umelana nemiphumela ye-insulin-ihomoni elawula ukuhamba kweshukela emangqamuzaneni akho-noma ayikhiqizi ngokwanele i-insulin ukuze igcine izinga elivamile le-glucose.
Okuvamile kubantu abadala, uhlobo lwe-2 lwesifo sikashukela luyaba nethonya kakhulu ezinganeni njengokwanda kwenani lomntwana . Akukho ukwelashwa kwesifo sikashukela sohlobo lwesibili, kodwa ungakwazi ukuphatha lesi simo ngokudla kahle, ukuzivocavoca nokugcina isisindo esinempilo. Uma ukudla nokuzivocavoca kunganele ukuphatha kahle ushukela wegazi lakho, ungase udinga imithi yesifo sikashukela noma ukwelashwa kwe-insulin.
Yeka kanjani i-Januvia isebenza
I-DPP-4 inesibopho sokuphula amaprotheni avuselela amangqamuzana akhiqiza i-insulini emva kokudla. Uma i-DPP-4 ingavinjelwa, ama-protein angasebenzisa ukukhishwa kwe-insulini isikhathi eside, ngaleyo ndlela anciphise izinga le-glucose egazini.
UJanuvia wabonisa imiphumela emihle ekuvivinyeni kwakamuva kokubili ngokuhambisana nezinye izidakamizwa, ezifana ne-metformin, futhi ngokwayo.
Inqunyelwe uhlobo lwesifo sikashukela kuphela.
Kwabanye abantu, ukudla, ukuzivocavoca, kanye nemithi ejwayelekile akufanelekile ukugcina amazinga e-glucose egazi ngezinga elihle. UJanuvia uye waphumelela ekuvivinyweni komtholampilo ekusizeni ukwehlisa uma izindlela zendabuko zinganele. Ukudla nokuzivocavoca kusekhona okunye okubalulekile ekuphathweni kwezokwelapha, noma kunjalo.
UJanuvia usebenza ngokukhulisa ukuvuselelwa kokukhiqizwa kwe-insulin. Ingozi ye- hypoglycemia ayinakwenzeka ngoba u-Januvia usebenza kuphela uma kudingeka. Isibonelo, uma kungekho glucose egazini, khona-ke akukho isenzo esivela ku-Januvia. Kodwa, emva kokudla lapho amazinga e-glucose ekhuphuka, uJanuvia uzosebenza ukuze anciphise lelo zinga.
Futhi, ososayensi bathole ukuthi kunengozi encane yokwehlisa isisindo ngoJanuwari, ngokungafani neminye imithi yesifo sikashukela yomlomo.
Okuqhamuka uma udla imishanguzo
Imiphumela emibi kakhulu ebikiwe ihlanganisa ukutheleleka okuphezulu kokuphefumula, umkhuhlane, kanye / noma ikhanda lokukhanda.
I-Januvia iqhutshwa ngezinso. Abantu abaye banciphisa umsebenzi we-renal kungadingeka ukuthi babe nomthamo wabo ka-Januvia oshintshwe udokotela wabo kumthamo ophansi. Umsebenzi wezintambo kufanele uhlolwe ngaphambi kokuthatha uJanuvia.
Umthombo:
Ukuphathwa kwe-US nokuDrug. I-FDA ivumela Ukwelashwa Okusha Kwesifo Sikashukela. Okthoba 2006.