Okwenza ama-Grapefruit nama-Statins Ungaxubeki

Ukusebenzisana Kungozidakamizwa Ezingozi, kuchazwe

Uma uthatha imithi ye-statin ukuphatha i-cholesterol ephakeme, kuye ngokuthi yikuphi okubekiwe, udokotela wakho noma umuthi wezokwelapha kungenzeka ugcizelele ukuthi akufanele udle izithelo zomvini noma uphuze ijusi lamagilebhisi ngenkathi usezidakamizweni. Ngenkathi lokho kungase kuzwakale kuyinqaba-kungani kungenjalo i-orange juice noma i-lemonade-kunesizathu esihle kakhulu sokususa le-citrus ethile.

I-Grapefruit ingasebenzisana neziqu ezithile ngezindlela ezingenza imithi ingasebenzi kahle futhi ingabangela neminye imiphumela engathandeki.

Okwenza ama-Grapefruit nama-Statins Ungaxubeki

Ngokomtholampilo, izitembu ziyaziwa ngokuthi i-HMG-CoA reductase inhibitors, isichazamazwi esichaza kahle ukuthi isebenza kanjani ekunciphiseni amazinga e-cholesterol-ngokuvimbela i-enzyme eyisihluthulelo ekukhiqizeni i-cholesterol emzimbeni obizwa ngokuthi i-HMG Co-A yokunciphisa. Izitatimende ziyi-anti-cholesterol ehlisa kakhulu imithi ngenxa yokuthi, ngaphezu kokuvimbela i-cholesterol, ithinta zonke izici zephrofayili yakho ye-lipid (i-lip-scrotein ephansi kakhulu, noma i- LDL ; i-lipoproteins ephakeme kakhulu, noma i- HDL ; ne- triglycerides ) ngendlela enhle .

I-grapefruit iqukethe i-bergamottin ebizwa ngokuthi i-bergamottin ehlangana nezinhlelo eziningi ze-enzyme emzimbeni, kuhlanganise ne-cytochrome P-450 ne-P-glycoprotein. Lezi zinhlelo ze-enzyme zinesibopho sokuphula phansi iziqu (nezinye izidakamizwa) zibe ngamakhemikhali umzimba ongasebenzisa kalula.

Uma udla i-grapefruit noma uphuza isiphuzo se-grapefruit lapho uthatha isithwathwa, i-bergamottin ingavimbela lezi zinhlelo ze-enzyme ukuthi zingabhidli izidakamizwa. Ngenxa yalokho, ingakwazi ukuqoqa ngobuningi emzimbeni wakho.

I-buildup of statins ingaba yingozi kakhulu, okungenzeka kubangele izinkinga zempilo ezinjengezinyimba ezinamandla zesibindi noma isimo esingavamile esibizwa ngokuthi i-rhabdomyolysis lapho izicubu zomzimba zihlahla khona, ukukhulula imicu ye-muscle ibe igazi elingalimaza izinso ngisho nokuholela ekulimazeni kwezinso.

Akuwona wonke ama-statin awahambisani namagilebhisi, kodwa lawo ahlanganisa, afaka:

Ezinye izitembu azibonwanga ukuthi zinenkinga uma zihlangene ne-grapefruit. Ososayensi bacabanga ukuthi lokhu kungenzeka ngoba abahlukunyezwa yizinhlelo ezifanayo ze-enzyme eziqukethe izidakamizwa. Zihlanganisa:

Ngisho neJuice encane ingahle ibe ningi kakhulu

Ucwaningo oluningi luye lwabonisa ukuthi kuthatha u-ounce owodwa kuphela osebenza ngejusi lamagilebhisi, noma i-grapefruit entsha ephelele, okubangela ukuba i-statins iqoqe emzimbeni. Ngakho-ke, uma uthatha i-Lipitor, i-Mevacor, noma i-Zocor kungcono ukucacisa ngokucacile imifino yamagilebhisi ngokuphelele. Uma uthanda ngempela i-grapefruit futhi uyamzonda umqondo wokuwunikela, khuluma nomhlinzeki wakho wezempilo ngokukushintshela kwesinye isifanekiso noma okungenani wehlise umthamo womuntu ozithathayo. Ngaleyo ndlela, uzokwazi ukujabulela i-grapefruit yakho futhi ungabhemi nemiphumela emibi. Kungase kube umqondo omuhle wokuqapha uma uthatha esinye isimiso ngokuthi ungadli i-grapefruit amahora ambalwa ngaphambi noma ngemuva kokuthatha le mithi.

> Imithombo:

> Dipiro JT, Talbert RL. I-Pharmacotherapy: Indlela Yokuthola Pathophysiological , 9th 2014.

> Lee JW, Morris JK, Wald NJ, et al. "IJupefruit Juice kanye nezitatimende." Am J Med 2016; 129: 26-29.

> IPhalamende le-Vaquero, iSanchez Muniz FJ, Redondo SJ et al. "Ukusebenzisana Okuyisidlo Sokudla Ngezidakamizwa Okuthinta Izici Zokuziphatha Nezimpahla Zama-Hypolipidaemic Statins." I-Nutr Hospital 2010; 25: 193-206.