Okudingeka Ukwazi NgeSkelaxin

I-Skelaxin (i-metaxalone) isetshenziselwa ukuphatha ubuhlungu be-muscle nokuqina kobuhlungu obubhekene nezimo ezibucayi, ezibuhlungu njenge-strain, sprains, noma ezinye ukulimala. Kuvame ukusetshenziselwa ukuhlanganiswa nokuphumula, ukwelashwa ngokomzimba.

Ngokwemvelo, ukubunjwa kunikezwa njenge-5 - [(3,5- (dimethylphenoxy) methyl] -2-oxazolidinone ngefomical formula C12H15N03 nesisindo samangqamuzana angu-221.25.

Indlela yokusebenza yalesi sidakamizwa ayizange ibonakale ngokucacile, kodwa ochwepheshe bakholelwa ukuthi lesi sidakamizwa sisebenza ngokuvimbela impulses yesisindo noma ukuzwa ubuhlungu ebuchosheni.

I-Skelaxin itholakale ngodokotela kuphela futhi inganikezwa iziguli ngezimo ezilandelayo:

Isilinganiso esinconywe

Umthamo ophakanyisiwe we-Skelaxin kubantu abadala nabantwana abaneminyaka engaphezu kwengu-12 ubudala eyodwa ye-800 mg tablet kane kathathu ngosuku. Kubalulekile ukuthi ungayithathi le mithi kunokuba udokotela wakho abekiwe. Imiphumela emibi yengozi ingenzeka uma uthatha okuningi.

I-Skelaxin igxila emathunjini amancane futhi igxiliswe ngesibindi futhi ixhunyiwe emcimbini njengemetabolite engaziwa.

Ubani ongafanelanga ukuthatha i-Skelaxin

Ngesikhathi iSkelaxin itholwe ukuthi iphephile ezigulini eziningi, iziguli ezithile akufanele zithathe.

Lokhu kufaka phakathi iziguli nganoma yikuphi ukuphathwa kwe-hypersensitivity kunoma yiziphi izingxenye zomuthi; labo abanomkhuba owaziwayo wezidakamizwa-induced, hemolytic, noma ezinye anemias; kanye nalabo abanomsebenzi wokuqamba amanga noma umsebenzi we-hepatic.

Ngaphezu kwalokho, iziguli ezidakwa utshwala kufanele zitshelwe ukuthi iSkelaxin ingathuthukisa imiphumela yotshwala nezinye izidakamizwa ze-CNS.

Kungase kuphazamise amakhono engqondo kanye / noma ngokomzimba okudingekayo ekusebenzeni imisebenzi enobungozi, njengemishini yokusebenza noma ukushayela imoto, ikakhulu uma isetshenziswe ngotshwala noma ezinye izidakamizwa ze-CNS.

Ukusetshenziswa okuphephile kwe-metaxalone akuzange kusungulwe ngokuphathelene nemiphumela emibi engenzeka ekuthuthukiseni ingane. Ngakho-ke, amaphilisi e-Skelaxin akufanele asetshenziswe kwabesifazane abakhulelwe noma abakhulelwe ikakhulukazi ngesikhathi sokukhulelwa kokuqala ngaphandle uma isahlulelo sodokotela kunenzuzo engaphezu kwezingozi ezikhona.

Ayaziwa ukuthi ngabe le mithi ifihlwe ubisi lomuntu. Njengomthetho jikelele, ukunakekelwa akufanele kwenziwe ngenkathi isiguli sisesidakamizweni njengoba izidakamizwa eziningi zixoshwa ebisi lomuntu. Ukusetshenziswa kwezingane, ukuphepha nokusebenza ezinganeni ezineminyaka engu-12 nangaphansi akukazanga.

Okuqhamuka uma udla imishanguzo

Nakuba kungavamile, ukusabela kwe-anaphylactoid kuye kwabikwa nge-Skelaxin. Izimpawu zokuphendula okubangayo zihlanganisa:

Ukusabela okuvame kakhulu ku-metaxalone kufaka:

> Umthombo:

Ukuphathwa Kwezokudla Nezidakamizwa zase-US, i-NDA 13-217 / S-036, ebuyekeziwe: Agasti, 2002